SCHEMBL20155262

SCHEMBL20155262

Cc1cc(N)ccc1Oc1ccc(C#N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.51
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
LRRK2 Q5S007 1/20 0.43
SLC6A4 P31645 1/20 0.42
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SCN9A Q15858 1/20 0.40
EPAS1 Q99814 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
MERTK Q12866 1/20 0.40
TEAD4 Q15561 1/20 0.39
MAP4K4 O95819 1/20 0.39
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20357553 0.87 AR (0.48) ARALDH1A1KDM4EUSP2SLC6A4
SCHEMBL2992329 0.86 ALDH1A1 (0.52) ALDH1A1KDM4ESLC6A4SMN1; SMN2TEAD4
SCHEMBL29688467 0.84 ALDH1A1 (0.55) ALDH1A1KDM4ESMN1; SMN2TEAD4
SCHEMBL1155719 0.84 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4
SCHEMBL31457276 0.84 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4
SCHEMBL3003478 0.84 ALDH1A1 (0.55) ALDH1A1KDM4ESMN1; SMN2TEAD4
SCHEMBL7020181 0.83 AR (0.46) ARALDH1A1KDM4EUSP2SLC6A4
SCHEMBL922953 0.83 AR (0.62) ARALDH1A1LRRK2SLC6A4SCN9A
SCHEMBL2748671 0.83 AR (0.51) ARALDH1A1KDM4EUSP2LRRK2
SCHEMBL27438050 0.82 AR (0.60) ARLRRK2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed