SCHEMBL20155404

SCHEMBL20155404

Cc1cc(N)c(C=N)cc1Oc1ccc(F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 10/20 0.40
MAP4K4 O95819 1/20 0.40
HSPB1 P04792 2/20 0.37
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
BRD4 O60885 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155521 0.83 EPAS1 (0.44) TRPA1MAP4K4HSPB1ALDH1A1
SCHEMBL20155430 0.82 TRPA1 (0.45) TRPA1MAP4K4HSPB1SLC6A2SLC6A4
SCHEMBL20160228 0.74 BRD4 (0.49) TRPA1MAP4K4HSPB1SLC6A2SLC6A4
SCHEMBL12181242 0.73 CYP3A4 (0.37) SLC6A2SLC6A4ALDH1A1
SCHEMBL10456772 0.71 TRPA1 (0.56) TRPA1MAP4K4HSPB1ALDH1A1
SCHEMBL2443815 0.71 EPAS1 (0.48) TRPA1MAP4K4HSPB1SLC6A2SLC6A4
SCHEMBL9658659 0.69 AR (0.47) TRPA1HSPB1SLC6A2SLC6A4SLC6A3
SCHEMBL1338646 0.69 KDM4E (0.55) TRPA1MAP4K4HSPB1SLC6A2SLC6A4
SCHEMBL22359718 0.69 NPC1 (0.38) ALDH1A1
SCHEMBL9658564 0.69 BRD4 (0.42) TRPA1SLC6A2SLC6A4SLC6A3BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed