SCHEMBL20155477

SCHEMBL20155477

Oc1ncc(Br)c2[nH]ncc12

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.37
AXL P30530 1/20 0.37
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
RET P07949 1/20 0.31
PI4KA P42356 1/20 0.31
XDH P47989 1/20 0.31
LRRK2 Q5S007 1/20 0.31
PI4K2B Q8TCG2 1/20 0.31
PI4K2A Q9BTU6 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
PTPN6 P29350 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30194269 1.00 NOS1 (0.37) NOS1AXLIDO1TDO2RET
SCHEMBL30550970 0.79 NOS1 (0.39) NOS1AXLIDO1TDO2RET
SCHEMBL20639279 0.79 NOS1 (0.39) NOS1AXLIDO1TDO2RET
SCHEMBL30515856 0.76 RET (0.47) NOS1AXLIDO1TDO2RET
SCHEMBL21579418 0.76 RET (0.47) NOS1AXLIDO1TDO2RET
SCHEMBL31260986 0.76 NOS1 (0.41) NOS1AXLIDO1TDO2RET
SCHEMBL25319103 0.72 PDPK1 (0.51) NOS1AXLRETPI4KAXDH
SCHEMBL24785354 0.72 AXL (0.37) NOS1AXL
SCHEMBL30966319 0.72 METAP2 (0.33) NOS1AXLRETPI4KAXDH
SCHEMBL25183087 0.72 METAP2 (0.33) NOS1AXLRETPI4KAXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed