SCHEMBL20155591

SCHEMBL20155591

Nc1cc(F)c(Nc2ccc(F)cc2F)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.44
IDO1 P14902 1/20 0.39
THRB P10828 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 4/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
ATM Q13315 1/20 0.36
MAP2K1 Q02750 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155425 0.80 SOS1 (0.46) SOS1IDO1THRBCYP2D6CYP2C19
SCHEMBL20155614 0.77 IDO1 (0.40) SOS1IDO1THRBALDH1A1GAA
SCHEMBL20155588 0.71 ALDH1A1 (0.37) SOS1CYP2D6CYP2C19ALDH1A1GAA
SCHEMBL17492772 0.71 SOS1 (0.48) SOS1THRBALDH1A1GAANPC1
SCHEMBL28924001 0.70 SOS1 (0.63) SOS1CYP2D6CYP2C19ALDH1A1GAA
SCHEMBL3607221 0.70 ALDH1A1 (0.44) SOS1CYP2D6CYP2C19ALDH1A1GAA
SCHEMBL15638643 0.69 ALDH1A1 (0.47) SOS1IDO1THRBCYP2D6CYP2C19
SCHEMBL20155496 0.69 SOS1 (0.42) SOS1IDO1THRBCYP2D6CYP2C19
SCHEMBL1662774 0.68 MAPK14 (0.41) SOS1CYP2D6CYP2C19ALDH1A1GAA
SCHEMBL16396266 0.68 SOS1 (0.48) SOS1CYP2D6CYP2C19ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed