SCHEMBL20155641

SCHEMBL20155641

O=[N+]([O-])c1ccc(Nc2ccc(Cl)cc2Cl)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.49
MAPT P10636 3/20 0.49
BCL6 P41182 2/20 0.49
BCOR Q6W2J9 2/20 0.49
ALDH1A1 P00352 2/20 0.49
TSHR P16473 2/20 0.49
MAPK1 P28482 2/20 0.49
MEN1 O00255 2/20 0.49
PKM P14618 2/20 0.49
HTT P42858 2/20 0.49
KMT2A Q03164 2/20 0.49
AURKA O14965 1/20 0.49
NPC1 O15118 1/20 0.49
PDPK1 O15530 1/20 0.49
JAK2 O60674 1/20 0.49
GMNN O75496 1/20 0.49
EGFR P00533 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155589 0.86 BCL6 (0.47) TDP1MAPTBCL6BCORALDH1A1
SCHEMBL20155624 0.84 BCL6 (0.60) TDP1MAPTBCL6BCORALDH1A1
Nitric Acid SCHEMBL11144683 0.77 TSHR (0.50) TDP1MAPTALDH1A1TSHRMAPK1
SCHEMBL11333871 0.77 BCL6 (0.63) TDP1MAPTBCL6BCORALDH1A1
SCHEMBL11492017 0.75 TSHR (0.62) TDP1MAPTALDH1A1TSHRMAPK1
SCHEMBL11741174 0.75 MAPK1 (0.53) TDP1MAPTBCL6BCORALDH1A1
SCHEMBL20155101 0.74 ALDH1A1 (0.47) TDP1ALDH1A1TSHRMAPK1HTT
SCHEMBL31252374 0.74 MAPT (0.68) TDP1MAPTBCL6BCORALDH1A1
SCHEMBL23779899 0.73 MAPT (0.53) TDP1MAPTBCL6BCORALDH1A1
SCHEMBL7606527 0.73 PDE7A (0.70) TSHRMAPK1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed