SCHEMBL20155646

SCHEMBL20155646

CC1(C)OB(c2cc(N)ccc2Nc2ccc(C(F)(F)F)cc2F)OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 6/20 0.36
PDGFRB P09619 1/20 0.34
KDR P35968 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KIF11 P52732 4/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
PDE2A O00408 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29074784 0.85 KDM4E (0.41) LIPEPDGFRBKDRALDH1A1MAPT
SCHEMBL20155117 0.85 ALDH1A1 (0.39) ALDH1A1MAPTKDM4EGAAL3MBTL1
SCHEMBL20155620 0.83 EGFR (0.37) LIPEPDGFRBKDRKMT2ACA1
SCHEMBL21904936 0.78 JAK2 (0.34) CA1CA2CA9EGFR
SCHEMBL20155461 0.77 TDO2 (0.38) LIPEALDH1A1MEN1GAAKMT2A
SCHEMBL29909454 0.76 PDE2A (0.39) LIPEPDGFRBKDRGAAPDE2A
SCHEMBL4108381 0.76 PDE2A (0.39) LIPEPDGFRBKDRGAAPDE2A
SCHEMBL20155119 0.75 MAPT (0.41) ALDH1A1MAPTKDM4EMEN1GAA
SCHEMBL44941 0.74 ALDH1A1 (0.38) LIPEALDH1A1MAPTKDM4EMEN1
SCHEMBL30990845 0.74 ALDH1A1 (0.38) LIPEALDH1A1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed