SCHEMBL20155693

SCHEMBL20155693

CCSNc1ccc(Oc2ccc(Cl)cc2F)c(C2=CN(C)C(=O)/C(=C/NC)C2=N)c1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.36
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
SCN9A Q15858 3/20 0.32
BRD2 P25440 1/20 0.30
BRD3 Q15059 1/20 0.30
BRDT Q58F21 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155445 0.93 BRD4 (0.39) BRD4BRD2BRD3BRDT
SCHEMBL20155073 0.90 BRD4 (0.38) BRD4SLC6A4KCNH2BRDT
SCHEMBL20155383 0.89 BRD4 (0.35) BRD4SLC6A2
SCHEMBL20155530 0.89 BRD4 (0.37) BRD4
SCHEMBL20155372 0.85 BRD4 (0.39) BRD4
SCHEMBL20155340 0.85 BRD4 (0.40) BRD4BRD2BRD3BRDT
SCHEMBL20155692 0.85 SLC6A2 (0.34) BRD4SLC6A2SLC6A4KCNH2SCN9A
SCHEMBL20155715 0.85 BRD4 (0.39) BRD4BRD2BRD3BRDT
SCHEMBL20155144 0.84 BRD4 (0.35) BRD4SCN9A
SCHEMBL20155690 0.84 BRD4 (0.38) BRD4BRD2BRD3BRDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed