SCHEMBL20155073

SCHEMBL20155073

CCSNc1ccc(Oc2ccc(Cl)cc2)c(C2=CN(C)C(=O)/C(=C/NC)C2=N)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.38
BRDT Q58F21 1/20 0.38
EP300 Q09472 1/20 0.33
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
KCNH2 Q12809 2/20 0.33
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
APEX1 P27695 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155693 0.90 BRD4 (0.36) BRD4BRDTSLC6A4KCNH2
SCHEMBL20155383 0.86 BRD4 (0.35) BRD4
SCHEMBL20155356 0.83 ALDH1A1 (0.34) BRD4BRDTEP300HTR2ASLC6A4
SCHEMBL20155530 0.81 BRD4 (0.37) BRD4
SCHEMBL20155144 0.81 BRD4 (0.35) BRD4
SCHEMBL20155340 0.77 BRD4 (0.40) BRD4BRDTEP300
SCHEMBL20155372 0.77 BRD4 (0.39) BRD4
SCHEMBL20155715 0.76 BRD4 (0.39) BRD4BRDTEP300
SCHEMBL20155690 0.76 BRD4 (0.38) BRD4BRDTEP300
SCHEMBL20155473 0.75 BRD4 (0.39) BRD4BRDTEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed