SCHEMBL20156064

SCHEMBL20156064

Oc1cn(O)nc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.47
GABRB2 P47870 5/20 0.47
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 4/20 0.41
MAPT P10636 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
BACE1 P56817 1/20 0.38
PTGIR P43119 1/20 0.37
HPGD P15428 2/20 0.37
USP2 O75604 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BCL2L1 Q07817 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALOX15 P16050 1/20 0.37
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21281611 0.78 KMT2A (0.44) ALDH1A1MAPTL3MBTL1MEN1KMT2A
SCHEMBL23400397 0.76 ALDH1A1 (0.57) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL23399527 0.75 KMT2A (0.43) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL23400421 0.73 RECQL (0.41) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL23400987 0.73 AURKA (0.37) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL23402101 0.71 PTGIR (0.44) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL23403188 0.70 ADORA3 (0.43) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL23399568 0.70 KMT2A (0.58) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL23398902 0.70 S1PR1 (0.45) ALDH1A1KDM4EMEN1KMT2APTGIR
SCHEMBL15135221 0.66 MEN1 (0.50) ALDH1A1KDM4EMAPTL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed