SCHEMBL20156248

SCHEMBL20156248

CC(C)(C)OC(=O)[C@@H](N)CNC(=O)/C(C=N)=C/NCCc1ccc2c(n1)NCCC2

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 14/20 0.44
ITGB6 P18564 9/20 0.44
CXCR4 P61073 6/20 0.43
ITGB3 P05106 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156055 0.88 ITGAV (0.47) ITGAVITGB6CXCR4ITGB3
SCHEMBL20156054 0.88 ITGAV (0.47) ITGAVITGB6CXCR4ITGB3
SCHEMBL20156298 0.84 ITGAV (0.57) ITGAVITGB6CXCR4ITGB3
SCHEMBL19825653 0.79 ITGAV (0.62) ITGAVITGB6ITGB3
SCHEMBL18104630 0.79 ITGAV (0.62) ITGAVITGB6ITGB3
SCHEMBL20156094 0.79 ITGAV (0.49) ITGAVITGB6CXCR4ITGB3
SCHEMBL20156009 0.78 CXCR4 (0.47) ITGAVITGB6CXCR4ITGB3
SCHEMBL20156008 0.78 ITGAV (0.53) ITGAVITGB6CXCR4ITGB3
SCHEMBL20156096 0.77 ITGAV (0.67) ITGAVITGB6ITGB3
SCHEMBL23912887 0.76 ITGAV (0.48) ITGAVITGB6CXCR4ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed