SCHEMBL23912887

SCHEMBL23912887

CCCCOC(=O)N[C@@H](CNC(=O)/C(C=N)=C/NCCc1ccc2c(n1)NCCC2)C(=O)OCC(C)C

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 18/20 0.48
ITGB6 P18564 11/20 0.48
ITGB3 P05106 7/20 0.45
CXCR4 P61073 2/20 0.40
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156096 0.81 ITGAV (0.67) ITGAVITGB6ITGB3ITGB1ITGA4
SCHEMBL20156298 0.80 ITGAV (0.57) ITGAVITGB6ITGB3CXCR4
SCHEMBL20156248 0.76 ITGAV (0.44) ITGAVITGB6ITGB3CXCR4
SCHEMBL20156054 0.76 ITGAV (0.47) ITGAVITGB6ITGB3CXCR4ITGB1
SCHEMBL20156009 0.75 CXCR4 (0.47) ITGAVITGB6ITGB3CXCR4
SCHEMBL20156297 0.75 ITGAV (0.51) ITGAVITGB6ITGB3ITGB1ITGA4
SCHEMBL20156008 0.73 ITGAV (0.53) ITGAVITGB6ITGB3CXCR4
SCHEMBL20156094 0.72 ITGAV (0.49) ITGAVITGB6ITGB3CXCR4
SCHEMBL24363128 0.69 ITGAV (0.61) ITGAVITGB6ITGB3ITGB1ITGA4
SCHEMBL21272499 0.69 ITGAV (0.53) ITGAVITGB6ITGB3ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed