SCHEMBL20156338

SCHEMBL20156338

N=C/C(=C\NCCc1ccc2c(n1)NCCC2)CNC[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 19/20 0.63
ITGB3 P05106 10/20 0.63
ITGB6 P18564 9/20 0.45
ITGB1 P05556 2/20 0.43
ITGA5 P08648 1/20 0.43
ITGA2B P08514 1/20 0.42
ITGA4 P13612 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156096 0.87 ITGAV (0.67) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL20156298 0.80 ITGAV (0.57) ITGAVITGB3ITGB6ITGA2B
SCHEMBL20141428 0.79 ITGAV (0.74) ITGAVITGB3ITGB6ITGB1ITGA4
SCHEMBL23912918 0.78 ITGB3 (0.56) ITGAVITGB3ITGB6ITGA2B
SCHEMBL6421342 0.78 ITGAV (1.00) ITGAVITGB3ITGB6
SCHEMBL6421344 0.78 ITGAV (1.00) ITGAVITGB3ITGB6
SCHEMBL20156337 0.77 ITGB3 (0.48) ITGAVITGB3ITGB6ITGA2B
SCHEMBL21272501 0.76 ITGAV (0.64) ITGAVITGB3ITGB6ITGA2B
SCHEMBL20139095 0.76 ITGAV (0.64) ITGAVITGB3ITGB6ITGA2B
SCHEMBL20156098 0.76 CXCR4 (0.47) ITGAVITGB3ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed