SCHEMBL20156337

SCHEMBL20156337

N=C/C(=C\NCCc1ccc2c(n1)NCCC2)CN(CCC(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 18/20 0.48
ITGAV P06756 18/20 0.48
ITGB5 P18084 6/20 0.41
ITGB6 P18564 4/20 0.41
ITGB8 P26012 3/20 0.41
CXCR4 P61073 2/20 0.41
ITGA2B P08514 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23912918 0.78 ITGB3 (0.56) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156338 0.77 ITGAV (0.63) ITGB3ITGAVITGB6ITGA2B
SCHEMBL20156335 0.76 TLR9 (0.32)
SCHEMBL20140239 0.75 ITGB3 (0.48) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156256 0.74 ITGB3 (0.52) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156008 0.73 ITGAV (0.53) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156098 0.73 CXCR4 (0.47) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20141252 0.72 ITGAV (0.55) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL23341168 0.71 ITGAV (0.65) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156094 0.70 ITGAV (0.49) ITGB3ITGAVITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed