SCHEMBL20157773

SCHEMBL20157773

COCc1ccc(N)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F11 P03951 1/20 0.40
LPL P06858 6/20 0.38
LIPG Q9Y5X9 6/20 0.38
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 2/20 0.34
UCHL1 P09936 1/20 0.34
CA2 P00918 2/20 0.32
ESR2 Q92731 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
PDK2 Q15119 1/20 0.31
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ANPEP P15144 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30526866 0.83 LPL (0.37) F11LPLLIPGLMNATP53
SCHEMBL15056893 0.83 LPL (0.37) F11LPLLIPGLMNATP53
SCHEMBL262723 0.83 LPL (0.37) F11LPLLIPGLMNATP53
SCHEMBL16971348 0.82 LPL (0.45) F11LPLLIPGUCHL1ESR2
SCHEMBL16971971 0.82 LPL (0.45) F11LPLLIPGUCHL1ESR2
SCHEMBL22768361 0.80 LPL (0.37) F11LPLLIPGLMNATP53
SCHEMBL17261770 0.80 LPL (0.37) F11LPLLIPGLMNATP53
SCHEMBL20157282 0.77 LIPG (0.37) F11LPLLIPGUCHL1CA2
SCHEMBL14714802 0.75 LPL (0.61) F11LPLLIPGCA2ESR2
SCHEMBL21550138 0.75 LPL (0.39) F11LPLLIPGUCHL1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed