SCHEMBL20157788

SCHEMBL20157788

Cn1cc(-c2ccccc2C(=O)c2ccc(Cl)cc2)c(C(CC(=O)OC(C)(C)C)NC(C)(C)C)cc1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
PTPRC P08575 2/20 0.37
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 3/20 0.34
P2RX3 P56373 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
MAPT P10636 3/20 0.32
NR4A1 P22736 1/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
MEN1 O00255 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 1/20 0.32
ALOX12 P18054 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362517 0.88 BRD4 (0.40) BRD4PTPRCKMT2AKDM4EP2RX3
SCHEMBL21362150 0.88 BRD4 (0.40) BRD4PTPRCKMT2AKDM4EP2RX3
SCHEMBL21362518 0.87 BRD4 (0.45) BRD4PTPRCKMT2AKDM4EP2RX3
SCHEMBL21362563 0.77 BRD4 (0.53) BRD4KMT2AKDM4EP2RX3MAPT
SCHEMBL21362113 0.76 PTPRC (0.30) PTPRC
SCHEMBL21362114 0.76 PTPRC (0.30) PTPRC
SCHEMBL20157810 0.76 BRD4 (0.46) BRD4KMT2AKDM4EPPARGPPARA
SCHEMBL21362559 0.76 BRD4 (0.52) BRD4KMT2AKDM4EP2RX3MAPT
SCHEMBL21362149 0.76 BRD4 (0.40) BRD4KMT2AKDM4EP2RX3ALDH1A1
SCHEMBL21352026 0.75 BRD4 (0.48) BRD4KMT2AKDM4EP2RX3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed