SCHEMBL21362517

SCHEMBL21362517

Cn1cc(-c2ccccc2C(=O)c2ccc(Cl)cc2)c([C@H](CC(=O)OC(C)(C)C)N[S@@+]([O-])C(C)(C)C)cc1=O

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.40
PTPRC P08575 2/20 0.34
KMT2A Q03164 1/20 0.32
CNR2 P34972 1/20 0.32
KDM4E B2RXH2 1/20 0.32
P2RX3 P56373 1/20 0.32
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362150 1.00 BRD4 (0.40) BRD4PTPRCKMT2ACNR2KDM4E
SCHEMBL21362113 0.89 PTPRC (0.30) PTPRC
SCHEMBL21362114 0.89 PTPRC (0.30) PTPRC
SCHEMBL20157788 0.88 BRD4 (0.43) BRD4PTPRCKMT2AKDM4EP2RX3
SCHEMBL21362149 0.87 BRD4 (0.40) BRD4KMT2ACNR2KDM4EP2RX3
SCHEMBL21362103 0.85 BRD4 (0.46) BRD4KMT2ACNR2KDM4EP2RX3
SCHEMBL21362518 0.83 BRD4 (0.45) BRD4PTPRCKMT2AKDM4EP2RX3
SCHEMBL21362230 0.80 BRD4 (0.39) BRD4
SCHEMBL21362229 0.80 BRD4 (0.39) BRD4
SCHEMBL9280622 0.77 BRD4 (0.37) BRD4PTPRCKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed