SCHEMBL20157930

SCHEMBL20157930

CCS(=O)(=O)Cc1ccc(C(=O)c2ccc(F)c(OC)c2)c(-c2cn(C)c(=O)cc2CN)c1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.37
MAPT P10636 2/20 0.33
CREBBP Q92793 2/20 0.33
POLB P06746 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.32
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21352099 0.85 BRD4 (0.34) BRD4MAPTCREBBPPOLB
SCHEMBL21362110 0.85 BRD4 (0.34) BRD4CREBBP
SCHEMBL20157926 0.85 BRD4 (0.37) BRD4MAPTCREBBPPOLB
SCHEMBL21352115 0.85 BRD4 (0.36) BRD4MAPTCREBBPPOLB
SCHEMBL21362728 0.81 BRD4 (0.36) BRD4MAPTCREBBPPOLB
SCHEMBL21354490 0.81 BRD4 (0.34) BRD4MAPTCREBBPPOLB
SCHEMBL21549998 0.80 BRD4 (0.35) BRD4MAP2K2MAP2K1
SCHEMBL21362158 0.79 BRD4 (0.34) BRD4CREBBP
SCHEMBL21362162 0.78 BRD4 (0.34) BRD4MAPTCREBBPPOLB
SCHEMBL21362088 0.78 BRD4 (0.42) BRD4MAPTMAP2K2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed