SCHEMBL21549998

SCHEMBL21549998

CCS(=O)(=O)Cc1ccc(C(=O)c2c(Cl)cc(F)cc2Cl)c(-c2cn(C)c(=O)cc2CN)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.35
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32
BAZ2B Q9UIF8 1/20 0.32
BAZ2A Q9UIF9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21564816 0.92 ALDH2 (0.35) BRD4BAZ2BBAZ2A
SCHEMBL21564957 0.85 ALDH2 (0.36) BRD4BAZ2BBAZ2A
SCHEMBL21564968 0.84 MAP2K2 (0.32) BRD4MAP2K2MAP2K1BAZ2BBAZ2A
SCHEMBL28468872 0.83 BRD4 (0.40) BRD4
SCHEMBL21362118 0.80 BRD4 (0.42) BRD4MAP2K2MAP2K1BAZ2BBAZ2A
SCHEMBL28470558 0.80 BRD4 (0.34) BRD4
SCHEMBL20157930 0.80 BRD4 (0.37) BRD4MAP2K2MAP2K1
SCHEMBL21550002 0.78 ALDH2 (0.34) BRD4BAZ2BBAZ2A
SCHEMBL21550003 0.78 ALDH2 (0.34) BRD4BAZ2BBAZ2A
SCHEMBL21564831 0.77 P2RX7 (0.34) BRD4MAP2K2MAP2K1BAZ2BBAZ2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed