SCHEMBL20157965

SCHEMBL20157965

Cc1ccc(C(=O)c2ccc(NC(=O)OC(C)(C)C)cc2-c2cn(C)c(=O)cc2[C@H](C)NN2C(=O)CCC2=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
RORC P51449 4/20 0.32
BCL2 P10415 1/20 0.32
BECN1 Q14457 1/20 0.32
BRD4 O60885 2/20 0.32
ACHE P22303 1/20 0.31
BACE1 P56817 1/20 0.31
MAPK14 Q16539 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CD274 Q9NZQ7 1/20 0.31
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158163 0.81
SCHEMBL21362490 0.80 MAPK14 (0.38) PRMT5WDR77MAPK14MEN1KMT2A
SCHEMBL20157833 0.77 BRD4 (0.31) BRD4
SCHEMBL20157861 0.76 EPHX2 (0.33) BRD4PPARG
SCHEMBL21362065 0.74 BRD4 (0.38) BRD4
SCHEMBL21362034 0.71 RAF1 (0.38) PRMT5WDR77RORCBRD4ACHE
SCHEMBL20157758 0.71 RAF1 (0.40) RORCBRD4ACHEBACE1RAF1
SCHEMBL20157708 0.71
SCHEMBL20157881 0.70 BRD4 (0.36) BRD4ALDH1A1
SCHEMBL28859608 0.70 MMP8 (0.39) CA12CA1CA9RORCBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed