SCHEMBL20158029

SCHEMBL20158029

CCCCCc1ccc(C(=O)c2ccc(C)cc2Cl)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 8/20 0.46
PPARA Q07869 2/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PLK3 Q9H4B4 2/20 0.44
PPARG P37231 1/20 0.42
KAT8 Q9H7Z6 2/20 0.42
RARB P10826 3/20 0.41
TRPM2 O94759 2/20 0.41
RARA P10276 1/20 0.39
RARG P13631 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362709 0.85 HPGD (0.42) NPC1RAB9A
SCHEMBL20157821 0.83 CYP4F2 (0.46) NPC1RAB9A
SCHEMBL21564940 0.80 HPGD (0.40) NPC1RAB9A
SCHEMBL20157822 0.80 HPGD (0.38) NPC1RAB9A
SCHEMBL20158005 0.79 HPGD (0.39) NPC1RAB9A
SCHEMBL21564804 0.78 CA1 (0.39) NPC1RAB9A
SCHEMBL11871709 0.77 PPARA (0.68) PLK1PPARAPLK3PPARGKAT8
SCHEMBL20504234 0.76 PPARA (0.70) PLK1PPARAPLK3PPARGKAT8
SCHEMBL8388149 0.76 PPARA (0.57) PPARAPPARGKAT8RARBRARA
SCHEMBL7139165 0.76 PPARA (0.54) PPARAPPARGKAT8RARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed