SCHEMBL20158005

SCHEMBL20158005

Cc1ccc(C(=O)c2ccc(CS(C)(=O)=O)cc2Br)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.39
RAB9A P51151 6/20 0.38
NPC1 O15118 5/20 0.38
PTPN1 P18031 1/20 0.36
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
ACHE P22303 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157822 0.89 HPGD (0.38) HPGDRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL21564804 0.89 CA1 (0.39) HPGDRAB9ANPC1MAPK13MAPK12
SCHEMBL21362178 0.86 NPC1 (0.41) HPGDRAB9ANPC1PTPN1MAPK13
SCHEMBL21362709 0.84 HPGD (0.42) HPGDRAB9ANPC1MAPTHTT
SCHEMBL20157821 0.84 CYP4F2 (0.46) HPGDRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL21362762 0.83 PTPN1 (0.33) HPGDPTPN1FLT1FLT4KDR
SCHEMBL20157951 0.83 MAPT (0.47) RAB9ANPC1PTPN1MAPTMAPK1
SCHEMBL21564940 0.81 HPGD (0.40) HPGDRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL21564702 0.79 CA12 (0.40) HPGDRAB9ANPC1MAPK13MAPK12
SCHEMBL20158029 0.79 PLK1 (0.46) RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed