SCHEMBL21362709

SCHEMBL21362709

CCc1ccc(C(=O)c2ccc(C)cc2Cl)c(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.42
RAB9A P51151 7/20 0.40
NPC1 O15118 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 3/20 0.40
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
PKM P14618 2/20 0.39
ALOX15 P16050 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157821 0.89 CYP4F2 (0.46) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL20157822 0.85 HPGD (0.38) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21564940 0.85 HPGD (0.40) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL20158029 0.85 PLK1 (0.46) RAB9ANPC1
SCHEMBL20158005 0.84 HPGD (0.39) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21564804 0.83 CA1 (0.39) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL23070442 0.79 HPGD (0.53) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21550127 0.79 SMN1; SMN2 (0.50) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21564740 0.78 MAPT (0.52) HPGDRAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21352079 0.77 HPGD (0.46) HPGDRAB9ANPC1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed