SCHEMBL20158053

SCHEMBL20158053

Cc1ccc(C(=O)c2ccc(C(C)S(=O)(=O)N(C)C(=O)OC(C)(C)C)cc2Br)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 2/20 0.36
MAPT P10636 3/20 0.34
HTT P42858 2/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
CNR2 P34972 3/20 0.32
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
KDM5A P29375 1/20 0.31
CA2 P00918 1/20 0.31
STAT5B P51692 1/20 0.30
ALDH1A1 P00352 2/20 0.30
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
GAA P10253 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362658 0.74 AAK1 (0.35) HTTCNR2ALDH1A1LMNA
SCHEMBL20158163 0.73
SCHEMBL21351900 0.73 CNR2 (0.35) CNR2CA2ALDH1A1LMNAGAA
SCHEMBL20157708 0.72
SCHEMBL20158166 0.69 MAPT (0.43) C5AR1MAPTHTTNPC1MAPK1
SCHEMBL20157584 0.68 CA12 (0.44) MAPTHTTNPC1MAPK1PPARG
SCHEMBL21352249 0.67 BACE1 (0.34) HTTCNR2ALDH1A1LMNA
SCHEMBL20157726 0.66 ACHE (0.34) MAPTHTTALDH1A1LMNA
SCHEMBL21564703 0.66 MAPT (0.33) MAPTHTTNPC1CNR2CA2
SCHEMBL11476383 0.66 MAPT (0.51) MAPTHTTNPC1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed