SCHEMBL20157726

SCHEMBL20157726

COc1cc(C(=O)c2ccc(CS(=O)(=O)N(C)C(=O)OC(C)(C)C)cc2Br)ccc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.34
ALDH1A1 P00352 1/20 0.34
BCHE P06276 5/20 0.34
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
PDF Q9HBH1 1/20 0.32
HTT P42858 1/20 0.31
CYP1A2 P05177 3/20 0.31
CYP2C19 P33261 3/20 0.31
CYP3A4 P08684 2/20 0.31
TSHR P16473 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP2D6 P10635 1/20 0.31
HPGD P15428 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158056 0.90 ACHE (0.35) ACHEALDH1A1BCHELMNAMTNR1A
SCHEMBL21362523 0.88 ACHE (0.33) ACHEALDH1A1BCHEMTNR1AMTNR1B
SCHEMBL20158011 0.82 CA12 (0.38) ACHEALDH1A1BCHELMNAMTNR1A
SCHEMBL20157485 0.80 ALDH1A1 (0.41) ACHEALDH1A1BCHEPDFCYP1A2
SCHEMBL20158058 0.80 ALDH1A1 (0.41) ACHEALDH1A1BCHELMNAPDF
SCHEMBL21564703 0.78 MAPT (0.33) ALDH1A1LMNASMN1; SMN2HTTMEN1
SCHEMBL21362793 0.76 PKM (0.49) ACHEALDH1A1BCHESMN1; SMN2CYP1A2
SCHEMBL20157609 0.76 ALDH1A1 (0.46) ACHEALDH1A1BCHECYP1A2CYP2C19
SCHEMBL21550462 0.76 NPC1 (0.36) ALDH1A1LMNAMEN1KMT2AHPGD
SCHEMBL20158078 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed