SCHEMBL20159103

SCHEMBL20159103

CC1CC(=O)N(C)N=C1c1ccc(N)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.41
CREBBP Q92793 2/20 0.41
GPR119 Q8TDV5 1/20 0.41
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
PIK3CD O00329 3/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
PIK3R1 P27986 5/20 0.35
PIK3CA P42336 5/20 0.35
MTOR P42345 5/20 0.35
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
SYK P43405 1/20 0.34
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
BRDT Q58F21 1/20 0.34
RICTOR Q6R327 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138813 0.82 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20142927 0.82 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159190 0.82 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL11393595 0.75 PDE4A (0.39) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL10549517 0.73 GPR119 (0.67) GPR119PDE4APDE4BPDE4CPDE4D
SCHEMBL22130329 0.73 PDE4B (0.36) PDE4APDE4BPDE4CPDE4DPDE3B
Cyanide SCHEMBL22130072 0.70 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9588042 0.69 PDE3B (0.69) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL11322162 0.69 PDE4A (0.51) CREBBPPDE4APDE4BPDE4CPDE4D
SCHEMBL11203913 0.69 PDE3B (0.63) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed