SCHEMBL20159634

SCHEMBL20159634

COc1cc(N2CC3C(N)C2[C@@H]3C)ccn1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.38
NR1H3 Q13133 3/20 0.38
LOX P28300 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
CYP17A1 P05093 3/20 0.35
SMARCA2 P51531 2/20 0.35
SMARCA4 P51532 2/20 0.35
CHRM4 P08173 3/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2D6 P10635 1/20 0.34
CHRM2 P08172 1/20 0.33
PROKR1 Q8TCW9 1/20 0.32
GRM2 Q14416 2/20 0.32
GAK O14976 1/20 0.32
ELOVL1 Q9BW60 1/20 0.31
ACVR2A P27037 1/20 0.31
TGFBR2 P37173 1/20 0.31
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159356 0.81 CHRM4 (0.32) LOXLOXL2CYP17A1CHRM4
SCHEMBL23504828 0.80
SCHEMBL20159687 0.76 NR1H2 (0.41) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL16685020 0.73 CHRM4 (0.47) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL19787604 0.72 CHRM4 (0.43) NR1H2NR1H3LOXLOXL2CYP17A1
Hydrochloric Acid SCHEMBL17077952 0.72 CHRM4 (0.47) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL21374488 0.71 PSEN1 (0.45) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL21069145 0.71 PSEN1 (0.45) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL21050448 0.71 PSEN1 (0.45) NR1H2NR1H3LOXLOXL2CYP17A1
SCHEMBL21050443 0.71 PSEN1 (0.45) NR1H2NR1H3LOXLOXL2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed