SCHEMBL20159356

SCHEMBL20159356

C[C@@H]1C2CN(c3ccnc(Cl)c3)C1C2N

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.32
LOX P28300 1/20 0.32
LOXL3 P58215 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
CYP17A1 P05093 4/20 0.32
MGLL Q99685 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159634 0.81 NR1H2 (0.38) CHRM4LOXLOXL2CYP17A1
SCHEMBL23504801 0.78 MMP2 (0.34)
SCHEMBL20159647 0.72 CHRNB2 (0.40) LOXLOXL3LOXL2CYP17A1
SCHEMBL20159670 0.72 LOX (0.32) CHRM4LOXLOXL3LOXL2CYP17A1
SCHEMBL20159656 0.69 CHRNA3 (0.39) CHRM4LOXLOXL3LOXL2CYP17A1
SCHEMBL18971107 0.68 CHRNB4 (0.38) CHRM4CYP17A1
SCHEMBL20031740 0.68 CHRM4 (0.38) CHRM4LOXLOXL3LOXL2CYP17A1
SCHEMBL20609194 0.68 CHRM4 (0.38) CHRM4LOXLOXL3LOXL2CYP17A1
SCHEMBL20609193 0.68 CHRM4 (0.38) CHRM4LOXLOXL3LOXL2CYP17A1
SCHEMBL18970901 0.68 CHRM4 (0.38) CHRM4LOXLOXL3LOXL2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed