SCHEMBL20160088

SCHEMBL20160088

CCOC(=O)Nc1cc(Br)cn2c(C)nnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 2/20 0.44
BRD4 O60885 2/20 0.44
BRD2 P25440 2/20 0.44
TRIM24 O15164 1/20 0.44
BRD1 O95696 1/20 0.44
TAF1 P21675 1/20 0.44
SMARCA4 P51532 1/20 0.44
BPTF Q12830 1/20 0.44
BRDT Q58F21 1/20 0.44
ATAD2 Q6PL18 1/20 0.44
PBRM1 Q86U86 1/20 0.44
TAF1L Q8IZX4 1/20 0.44
CREBBP Q92793 1/20 0.44
KAT2B Q92831 1/20 0.44
CECR2 Q9BXF3 1/20 0.44
BRD9 Q9H8M2 1/20 0.44
BRD7 Q9NPI1 1/20 0.44
BAZ2A Q9UIF9 1/20 0.44
BRPF3 Q9ULD4 1/20 0.44
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16267911 0.84 RXFP1 (0.36) BRD4BRD2ATAD2CREBBPBRD9
SCHEMBL17679224 0.84 BRD9 (0.52) BRD4BRD2CREBBPBRD9BRD3
SCHEMBL21227653 0.82 CYP1A2 (0.41) BRD4BRD2CREBBPCYP1A2BRD3
SCHEMBL20160220 0.73 BRPF1 (0.58) BRPF1BRD4BRD2TRIM24BRD1
SCHEMBL20160351 0.72 BRPF1 (0.57) BRPF1BRD4BRD2TRIM24BRD1
SCHEMBL31287064 0.70 ALDH1A1 (0.54) CYP1A2CYP2C9CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL16268761 0.69 MEN1 (0.36) BRD4KMT2AMEN1
SCHEMBL20160338 0.68 BRD4 (0.42) BRD4CREBBPCECR2SMN1; SMN2ALDH1A1
SCHEMBL15834999 0.68 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL1585857 0.68 CYP1A2 (0.48) CYP1A2CYP2C9CYP2C19SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed