SCHEMBL20160255

SCHEMBL20160255

Nc1ccc(Oc2ccc(F)cc2P)c(-c2ccc3c(c2)C(=O)NC3=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.40
MAOA P21397 3/20 0.38
MAOB P27338 3/20 0.38
BRD4 O60885 7/20 0.37
GRM5 P41594 2/20 0.36
TDP2 O95551 2/20 0.35
MAPK14 Q16539 1/20 0.34
CHEK1 O14757 2/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
MEN1 O00255 1/20 0.32
PRKD3 O94806 1/20 0.32
EGFR P00533 1/20 0.32
PRKCG P05129 1/20 0.32
PRKCB P05771 1/20 0.32
MAPT P10636 1/20 0.32
SRC P12931 1/20 0.32
PRKCA P17252 1/20 0.32
PRKCH P24723 1/20 0.32
PRKCI P41743 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159919 0.88 BRD4 (0.47) ATMMAOAMAOBBRD4GRM5
SCHEMBL20160256 0.81 BRD4 (0.38) ATMMAOAMAOBBRD4GRM5
SCHEMBL372282 0.70 ATM (0.58) ATMMAOAMAOBGRM5TDP2
Hydrochloric Acid SCHEMBL14890696 0.68 ATM (0.56) ATMMAOAMAOBGRM5TDP2
SCHEMBL20159920 0.68 BRD4 (0.48) ATMBRD4MAPK14
SCHEMBL29535893 0.67 GRM5 (0.63) MAOAMAOBGRM5TDP2MEN1
SCHEMBL1953630 0.67 GRM5 (0.63) MAOAMAOBGRM5TDP2MEN1
SCHEMBL15549928 0.66 BRD4 (0.53) BRD4
SCHEMBL28475420 0.65 BRD4 (0.47) BRD4MAPK14
SCHEMBL20160288 0.65 BRD4 (0.46) BRD4MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed