SCHEMBL20159920

SCHEMBL20159920

Nc1ccc(Oc2ccc(F)cc2F)c(-c2cccc3c2C(=O)NC3=O)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.48
MAPK14 Q16539 1/20 0.41
TRPA1 O75762 1/20 0.40
ATM Q13315 1/20 0.38
HSPB1 P04792 1/20 0.37
STK10 O94804 1/20 0.36
SLK Q9H2G2 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
BRDT Q58F21 1/20 0.36
CREBBP Q92793 1/20 0.36
CASP3 P42574 1/20 0.36
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160282 0.80 BRD4 (0.49) BRD4BRD2BRD3BRDT
SCHEMBL20159919 0.80 BRD4 (0.47) BRD4MAPK14ATM
SCHEMBL11307123 0.78 WEE1 (0.51) ATMSTK10SLKCASP3
SCHEMBL21904799 0.74 BRD4 (0.50) BRD4MAPK14TRPA1BRD2BRD3
SCHEMBL29845843 0.71 BRD4 (0.46) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL16654848 0.71 BRD4 (0.50) BRD4MAPK14TRPA1BRD2BRD3
SCHEMBL16650144 0.70 BRD4 (0.55) BRD4
SCHEMBL19930712 0.70 BRD4 (0.68) BRD4
SCHEMBL262473 0.69 GSK3B (0.50) ATMSTK10SLKCASP3
SCHEMBL21904906 0.68 BRD4 (0.66) BRD4MAPK14TRPA1BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed