SCHEMBL20160294

SCHEMBL20160294

CCSN(CC1CC1)c1ccc(Oc2ccc(F)cc2F)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 17/20 0.43
EPAS1 Q99814 1/20 0.39
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HSPB1 P04792 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159925 0.82 BRD4 (0.62) BRD4EPAS1
SCHEMBL20159849 0.77 BRD4 (0.45) BRD4
SCHEMBL20159993 0.69 BRD4 (0.62) BRD4
SCHEMBL15068022 0.68 EPAS1 (0.46) BRD4EPAS1HSPB1
SCHEMBL20154947 0.67 EPAS1 (0.45) BRD4EPAS1SLC6A2SLC6A4SLC6A3
SCHEMBL20160276 0.67 EPAS1 (0.45) BRD4EPAS1SLC6A2SLC6A4HSPB1
SCHEMBL16650857 0.66 EPAS1 (0.67) BRD4EPAS1HSPB1
SCHEMBL20384507 0.66 EPAS1 (0.47) EPAS1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL20384414 0.66 EPAS1 (0.55) EPAS1SLC6A2SLC6A4SLC6A3HSPB1
SCHEMBL20443103 0.65 HTR1A (0.38) BRD4EPAS1HTR1ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed