SCHEMBL20160668

SCHEMBL20160668

Cc1cnc(CN2CCN(C)CC2)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.39
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
CHKA P35790 2/20 0.38
AXL P30530 3/20 0.38
MC4R P32245 1/20 0.38
KDM4A O75164 1/20 0.36
KDM4B O94953 1/20 0.36
KDM5C P41229 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
MPO P05164 1/20 0.36
LMNA P02545 1/20 0.36
TNIK Q9UKE5 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160907 0.83 NPC1 (0.44) LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL20160565 0.83 TNKS (0.41) TNKSPARP1TNKS2CHKAAXL
SCHEMBL15214350 0.77 ALDH1A1 (0.39) LMNAKDM4EALDH1A1SMN1; SMN2GRIN1
SCHEMBL15198047 0.75 HRH3 (0.46) KDM4ESMN1; SMN2GRIN1GRIN2B
SCHEMBL12767186 0.75 BCHE (0.38) TNKSPARP1TNKS2ALDH1A1TLR7
SCHEMBL12727211 0.74 ALOX5AP (0.39) TLR7GRIN1GRIN2B
SCHEMBL18713006 0.73 TNKS (0.50) TNKSPARP1TNKS2CHKAMC4R
SCHEMBL20160541 0.73 TNKS (0.45) TNKSPARP1TNKS2CHKAMC4R
SCHEMBL21937884 0.73 SMN1; SMN2 (0.40) CHKAAXLMC4RKDM4AKDM4B
SCHEMBL20261166 0.72 CCR1 (0.37) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed