SCHEMBL20160541

SCHEMBL20160541

Cc1cnc(CN2CCN(C)CC2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.45
PARP1 P09874 1/20 0.45
TNKS2 Q9H2K2 1/20 0.45
MC4R P32245 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
GAA P10253 1/20 0.43
LMNA P02545 2/20 0.42
CHKA P35790 2/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 4/20 0.39
PTPN1 P18031 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
CA2 P00918 1/20 0.38
NCF1 P14598 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21551702 0.83 KDM4E (0.45) MC4RSMN1; SMN2GAALMNACHKA
SCHEMBL13923299 0.80 MC4R (0.52) TNKSPARP1TNKS2MC4RSMN1; SMN2
SCHEMBL15219267 0.79 CXCR4 (0.45) TNKSPARP1TNKS2LMNAPTPN1
SCHEMBL19145771 0.79 SMN1; SMN2 (0.47) SMN1; SMN2GAAKDM4EALDH1A1NPC1
SCHEMBL27360423 0.78 MC4R (0.46) MC4RSMN1; SMN2GAALMNACHKA
SCHEMBL26844932 0.78 ALDH1A1 (0.51) TNKSPARP1TNKS2SMN1; SMN2DRD4
SCHEMBL20322780 0.78 HDAC6 (0.43) MC4RLMNACHKAKDM4EALDH1A1
SCHEMBL12513 0.77 LTA4H (0.45) MC4RSMN1; SMN2GAALMNACHKA
SCHEMBL21604387 0.75 TNKS (0.37) TNKSPARP1TNKS2ALDH1A1
SCHEMBL9607176 0.75 GAA (0.38) MC4RSMN1; SMN2GAALMNACHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed