SCHEMBL20162086

SCHEMBL20162086

Cc1cn2ccc(O)nc2n1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
PDE10A Q9Y233 4/20 0.35
GRM5 P41594 2/20 0.33
NPC1 O15118 2/20 0.30
GAA P10253 2/20 0.30
KMT2A Q03164 2/20 0.30
POLB P06746 1/20 0.30
GFER P55789 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10143645 0.83 PDE10A (0.38) HDAC1PDE10AGRM5NPC1GAA
SCHEMBL17626629 0.76 SUV39H2 (0.44) HDAC1PDE10AGRM5ADORA3ADORA2A
SCHEMBL12343964 0.73 PDE8B (0.35) HDAC1PDE10AGRM5NPC1POLB
SCHEMBL12341046 0.73 PDE10A (0.33) HDAC1PDE10AGRM5NPC1GAA
SCHEMBL20344162 0.72 PDE10A (0.33) HDAC1PDE10A
SCHEMBL17285646 0.72 HDAC1 (0.35) HDAC1PDE10A
SCHEMBL25124896 0.68 PDE10A (0.35) PDE10ANPC1GAAKMT2AKDM4E
SCHEMBL12402544 0.68 PDE10A (0.35) HDAC1PDE10ANPC1GAAKMT2A
SCHEMBL25044484 0.68 PDE8B (0.39) PDE10ANPC1GAAKMT2AADORA3
SCHEMBL25124961 0.67 PDE10A (0.43) PDE10ANPC1GAAKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323821-A1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS Pfizer Inc (US) 2018-05-23 EP disclosed