SCHEMBL25044484

SCHEMBL25044484

Cc1ccn2cc(N)nc2n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE8B O95263 1/20 0.39
NOS3 P29474 3/20 0.39
NOS2 P35228 3/20 0.39
SUV39H2 Q9H5I1 6/20 0.38
PIK3CG P48736 1/20 0.36
PDE10A Q9Y233 4/20 0.35
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
PARP1 P09874 1/20 0.33
NOS1 P29475 2/20 0.30
RAB9A P51151 2/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17626629 0.84 SUV39H2 (0.44) PDE8BNOS3NOS2SUV39H2PDE10A
SCHEMBL10143645 0.83 PDE10A (0.38) PDE8BPDE10AADORA3ADORA2APARP1
SCHEMBL15101433 0.75 RAB9A (0.59) PDE10AADORA2ARAB9AKMT2AKDM4E
SCHEMBL17275572 0.71 PDE10A (0.63) PDE10AADORA2ARAB9AKMT2AKDM4E
SCHEMBL20162086 0.68 HDAC1 (0.35) PDE10AADORA3ADORA2ARAB9AKMT2A
SCHEMBL7314198 0.68 HTT (0.39) KDM4EALDH1A1
SCHEMBL6102107 0.67 ALDH1A1 (0.39) RAB9AKMT2AKDM4EMEN1NPC1
SCHEMBL15101432 0.67 PDE10A (0.45) PDE10ARAB9AKMT2AKDM4EMEN1
SCHEMBL12343964 0.65 PDE8B (0.35) PDE8BPDE10ARAB9AKDM4ENPC1
SCHEMBL12341046 0.65 PDE10A (0.33) PDE10ARAB9AKMT2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023018648-A1 PHENOL DERIVATIVES FOR USE IN THE MODULATION OF BRM GENENTECH, INC. (US) 2023-02-16 WO disclosed