SCHEMBL20162412

SCHEMBL20162412

CC(C)(C)OC(=O)N1CCCC1c1ccccc1-c1cncn1C1CC1.O=C(Oc1ccc(Cl)cc1)N1CCCC1c1ccccc1-c1cncn1CCc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 11/20 0.40
PIM1 P11309 1/20 0.39
MARK3 P27448 1/20 0.39
MAP4K2 Q12851 1/20 0.39
CAMK2B Q13554 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2B6 P20813 1/20 0.36
AADAT Q8N5Z0 3/20 0.35
CYP11B2 P19099 1/20 0.34
APP P05067 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
SLC6A2 P23975 1/20 0.33
HRH2 P25021 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16730873 0.91 AADAT (0.41) IDO1CYP3A4CYP2D6CYP2B6AADAT
SCHEMBL16730872 0.88 IDO1 (0.44) IDO1PIM1MARK3MAP4K2CAMK2B
SCHEMBL16730871 0.80 PIM1 (0.55) IDO1PIM1MARK3MAP4K2CAMK2B
SCHEMBL16730879 0.78 IDO1 (0.42) IDO1CYP3A4CYP2D6CYP2B6CYP11B2
SCHEMBL20162457 0.77 IDO1 (0.42) IDO1CYP3A4CYP2D6CYP2B6CYP11B2
SCHEMBL16730887 0.77 IDO1 (0.42) IDO1CYP3A4CYP2D6CYP2B6CYP11B2
SCHEMBL18128804 0.75 FKBP1A (0.44) IDO1CYP3A4CYP2D6CYP2B6AADAT
SCHEMBL16719008 0.75 FKBP1A (0.44) IDO1CYP3A4CYP2D6CYP2B6AADAT
SCHEMBL18134517 0.75 IDO1 (0.47) IDO1PIM1MARK3MAP4K2CAMK2B
SCHEMBL16730949 0.75 IDO1 (0.47) IDO1PIM1MARK3MAP4K2CAMK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP claimed