SCHEMBL2016433

SCHEMBL2016433

NCCc1cc(F)c2ccnnc2c1-c1cccc(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.43
BCL2 P10415 1/20 0.38
PIK3CD O00329 1/20 0.36
NOTUM Q6P988 1/20 0.34
KDM4E B2RXH2 1/20 0.33
SYK P43405 1/20 0.33
HTR2A P28223 2/20 0.33
MPO P05164 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
HTR1A P08908 1/20 0.32
KMT2A Q03164 1/20 0.32
GCGR P47871 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
DHODH Q02127 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12491178 0.89 BCL2 (0.47) TAAR1BCL2PIK3CDNOTUMKDM4E
SCHEMBL2016661 0.89 PIK3CD (0.36) TAAR1BCL2PIK3CDNOTUMKDM4E
SCHEMBL2014788 0.84 TAAR1 (0.43) TAAR1PIK3CDKDM4ESYKHTR2A
Trifluoroacetic Acid SCHEMBL2012078 0.81 BCL2 (0.41) TAAR1BCL2PIK3CDCYP3A4GRIN2B
SCHEMBL12403232 0.79 BCL2 (0.48) TAAR1BCL2PIK3CDNOTUMKDM4E
SCHEMBL2015599 0.78 BCL2 (0.36) TAAR1BCL2PIK3CDHTR2AMPO
SCHEMBL2016719 0.78 PIK3CD (0.47) TAAR1BCL2PIK3CDSYK
SCHEMBL2019261 0.77 PIK3CD (0.44) BCL2PIK3CDNOTUMKDM4ECYP17A1
SCHEMBL2016428 0.77 BCL2 (0.48) TAAR1BCL2PIK3CDNOTUMKDM4E
SCHEMBL12631928 0.76 PIK3CD (0.47) TAAR1BCL2PIK3CDNOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed