SCHEMBL2016440

SCHEMBL2016440

CCn1c(COC(=O)c2nc(Cl)c(N)nc2N)[n+](CC)c2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 4/20 0.37
HPGD P15428 4/20 0.37
HSD17B10 Q99714 4/20 0.37
GAA P10253 2/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SCNN1A P37088 4/20 0.36
DRD5 P21918 1/20 0.36
SCNN1B P51168 1/20 0.36
SCNN1G P51170 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
GRM5 P41594 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2D6 P10635 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL2024368 0.99 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12635739 0.92 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12636678 0.91 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12635726 0.91 APOBEC3A (0.39) ALDH1A1KDM4EHPGDHSD17B10GAA
Bromide SCHEMBL2053994 0.91 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12635761 0.91 APAF1 (0.35) ALDH1A1KDM4EHPGDHSD17B10GAA
Bromide SCHEMBL2049875 0.90 APOBEC3A (0.39) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12635737 0.89 APAF1 (0.41) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12636679 0.89 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL12636337 0.88 ADORA2A (0.37) ALDH1A1KDM4EHPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO claimed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed