SCHEMBL20168666

SCHEMBL20168666

C=CCC[C@H](Cc1ccc(C(=O)OC(C)(C)C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.38
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
SMO Q99835 1/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CACNA1B Q00975 5/20 0.35
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179138 1.00 SLC7A5 (0.38) SLC7A5THRATHRBCA12CA1
SCHEMBL20179148 0.92 CA12 (0.40) CA12CA1CA2CA9CA14
SCHEMBL20168531 0.92 CA12 (0.40) CA12CA1CA2CA9CA14
SCHEMBL20168301 0.91 CYP4F2 (0.44) THRATHRBCA12CA1CA2
SCHEMBL20179181 0.91 CYP4F2 (0.44) THRATHRBCA12CA1CA2
SCHEMBL20179248 0.86 SLC7A5 (0.56) SLC7A5MEN1CYP3A4KMT2ATDP1
SCHEMBL21578054 0.85 SLC7A5 (0.39) SLC7A5THRATHRBCA12CA1
SCHEMBL20179262 0.82 SLC7A5 (0.49) SLC7A5FOLH1PRSS1
SCHEMBL20168730 0.82 CPA3 (0.46) SLC7A5CA12CA1CA2CA9
SCHEMBL23833858 0.80 REN (0.44) TDP1L3MBTL1FOLH1MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094334-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-05-24 WO disclosed