SCHEMBL20169140

SCHEMBL20169140

Cc1ncc(-c2ccc(NC(=O)c3cc(F)cc(F)c3)cc2)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.48
PTPN11 Q06124 2/20 0.48
PTPN6 P29350 1/20 0.46
BACE1 P56817 1/20 0.45
AURKA O14965 2/20 0.45
AURKB Q96GD4 1/20 0.45
SCN9A Q15858 1/20 0.45
MAOB P27338 1/20 0.44
DGAT1 O75907 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GRM5 P41594 1/20 0.43
GSK3B P49841 1/20 0.43
KIT P10721 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26304040 0.87 BACE1 (0.50) BACE1SCN9AGRM5
SCHEMBL13655235 0.85 SCN9A (0.62) PTPN1PTPN11PTPN6BACE1AURKA
SCHEMBL6885895 0.74 PTPN1 (0.64) PTPN1PTPN11PTPN6BACE1NPC1
SCHEMBL7483325 0.73 CYP2A6 (0.53) BACE1NPC1RAB9ASMN1; SMN2GSK3B
SCHEMBL13655269 0.72 SCN9A (0.59) BACE1SCN9AKIT
SCHEMBL23812448 0.71 SCN9A (0.63) PTPN1PTPN11SCN9ANPC1RAB9A
SCHEMBL23812447 0.70 SCN9A (0.62) AURKASCN9AMAOB
SCHEMBL23326698 0.70 NQO2 (0.70) PTPN1NPC1RAB9ASMN1; SMN2
SCHEMBL677476 0.69 MEN1 (0.67) PTPN1NPC1RAB9ASMN1; SMN2
SCHEMBL23352870 0.68 TRPV1 (0.67) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975857-B2 Inhibition of bacterial biofilms with imidazole-phenyl derivatives NORTH CAROLINA STATE UNIVERSITY (US) 2018-05-22 US disclosed