SCHEMBL20169993

SCHEMBL20169993

O=C(Nc1cc2c(cc1F)CNCC2)c1cn(CC2C=C(F)C(F)=C(F)C2)cn1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 2/20 0.33
HDAC2 Q92769 2/20 0.32
HDAC1 Q13547 1/20 0.32
S1PR1 P21453 2/20 0.31
MELK Q14680 1/20 0.31
GPR6 P46095 1/20 0.30
WNT1 P04628 2/20 0.30
GSK3B P49841 2/20 0.30
DYRK1A Q13627 2/20 0.30
CLK2 P49760 1/20 0.30
CLK3 P49761 1/20 0.30
ATR Q13535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162149 0.78 MAP3K5 (0.34) MAP3K5HDAC2HDAC1S1PR1MELK
SCHEMBL21533383 0.77 WNT1 (0.35) MAP3K5MELKWNT1GSK3BDYRK1A
SCHEMBL20367451 0.77 HDAC1 (0.38) MAP3K5HDAC2HDAC1S1PR1MELK
SCHEMBL20162140 0.67 WNT1 (0.38) MAP3K5WNT1GSK3BDYRK1ACLK2
SCHEMBL20162145 0.66 SCD (0.39) MAP3K5WNT1GSK3BDYRK1ACLK2
SCHEMBL20162167 0.65 MELK (0.46) S1PR1MELK
Hydrochloric Acid SCHEMBL20162129 0.64 MELK (0.45) S1PR1MELK
SCHEMBL20162148 0.63 RBP4 (0.34) MAP3K5GPR6
SCHEMBL21518083 0.61 OGA (0.37)
SCHEMBL26107113 0.61 MELK (0.39) MAP3K5MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323809-A1 BICYCLIC HETEROCYCLIC AMIDE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-05-23 EP disclosed