SCHEMBL20170435

SCHEMBL20170435

O=S(=O)(NCc1ccccc1-c1cncn1CCc1ccc(F)cc1)c1cnc(N2CCN3CCCC3C2)s1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
KCNH2 Q12809 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719021 0.89
SCHEMBL20170514 0.87 KCNH2 (0.32) ATRKCNH2HRH3
SCHEMBL18128794 0.84 POLB (0.34) KCNH2
SCHEMBL20169605 0.83 CYP11B2 (0.33) ATR
SCHEMBL20170406 0.83 CYP11B2 (0.33) ATR
SCHEMBL20170477 0.80 SCN9A (0.31)
SCHEMBL16730869 0.80 CYP11B1 (0.35)
SCHEMBL16730866 0.79 CYP11B1 (0.35)
SCHEMBL16719037 0.76 HSP90AA1 (0.32)
SCHEMBL16719040 0.76 HSP90AA1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed