SCHEMBL20170477

SCHEMBL20170477

O=S(=O)(c1cnc(N2CCN3CCCC3C2)s1)N1CCc2c(cccc2-c2cncn2CCc2ccc(F)cc2)C1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
HTR6 P50406 1/20 0.31
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719019 0.90 SCN9A (0.31) SCN9A
SCHEMBL16719028 0.88 SCN9A (0.39) SCN9AP2RX3
SCHEMBL16718973 0.85 ADRA2C (0.30)
SCHEMBL20169617 0.85 ADRA2C (0.30)
SCHEMBL20170445 0.85 PRCP (0.35) SCN9ADRD2DRD3HTR6ALOX5AP
SCHEMBL20170406 0.82 CYP11B2 (0.33) ALOX5APFEN1
SCHEMBL20169605 0.82 CYP11B2 (0.33) ALOX5APFEN1
SCHEMBL16718968 0.82 DRD3 (0.35) SCN9ADRD2DRD3HTR6P2RX3
SCHEMBL16731026 0.80
SCHEMBL20169608 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed