SCHEMBL20170504

SCHEMBL20170504

CCc1ccc(CCn2cncc2-c2cccc3c2CNCC3)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRCP P42785 1/20 0.41
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
IDO1 P14902 1/20 0.36
PNMT P11086 2/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
HRH3 Q9Y5N1 1/20 0.33
P2RX7 Q99572 1/20 0.32
HTR7 P34969 2/20 0.32
HTR6 P50406 2/20 0.32
HTR1A P08908 1/20 0.32
SCN9A Q15858 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16731021 0.90 PRCP (0.41) PRCPHSP90AA1HSP90AB1PNMTCYP11B1
SCHEMBL16730831 0.82 CYP11B1 (0.39) HSP90AA1HSP90AB1IDO1CYP11B1CYP11B2
SCHEMBL16730944 0.81 CYP11B1 (0.41) HSP90AA1HSP90AB1IDO1CYP11B1CYP11B2
SCHEMBL20170503 0.74 PRCP (0.51) PRCPIDO1PNMTHRH3
SCHEMBL16730894 0.70 KCNH2 (0.37) HSP90AA1HSP90AB1CYP11B1CYP11B2HTR7
SCHEMBL16730963 0.69 ASIC3 (0.44) CYP11B1CYP11B2
SCHEMBL16730822 0.66 ABHD6 (0.39) IDO1CYP11B1CYP11B2SCN9A
SCHEMBL16730943 0.65 CYP11B1 (0.47) IDO1CYP11B1CYP11B2P2RX7HTR7
SCHEMBL26548216 0.65 PRCP (0.60) PRCPPNMTHTR6IRAK4
SCHEMBL16730958 0.64 HTR2C (0.38) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed