SCHEMBL20170712

SCHEMBL20170712

COc1ccc2c(c1OCc1ccccc1)C1(C)CC(=O)[C@H](C)CC1[C@@H](N)C2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
AGTR2 P50052 10/20 0.38
AGTR1 P30556 2/20 0.38
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
KDM1A O60341 5/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18458091 0.76 OPRM1 (0.36) MEN1HTTKMT2AAGTR2AGTR1
SCHEMBL21202021 0.70 MEN1 (0.36) MEN1HTTKMT2ABRD4CREBBP
SCHEMBL12013639 0.67 OPRM1 (0.36) MEN1HTTKMT2AAGTR2AGTR1
SCHEMBL12646217 0.67 OPRM1 (0.36) MEN1HTTKMT2AAGTR2AGTR1
SCHEMBL12013637 0.67 OPRM1 (0.51)
SCHEMBL27924335 0.67 OPRM1 (0.51)
SCHEMBL22058857 0.66 OPRM1 (0.37) MEN1HTTKMT2AAGTR2AGTR1
SCHEMBL18458090 0.66 GAA (0.44) MEN1KMT2AAGTR2AGTR1BCHE
SCHEMBL18474049 0.64 MEN1 (0.37) MEN1HTTKMT2AAGTR2AGTR1
SCHEMBL21300617 0.63 BCHE (0.67) BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed