SCHEMBL20171548

SCHEMBL20171548

CC(=O)c1ccc2c(C)c(OC3CCC(C(F)(F)F)CC3)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 8/20 0.52
LPAR1 Q92633 1/20 0.42
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
KDM2B Q8NHM5 4/20 0.39
SCN9A Q15858 3/20 0.38
RORC P51449 1/20 0.37
CYP2A6 P11509 1/20 0.36
APP P05067 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17057724 1.00 ENPP2 (0.52) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL17045111 0.88 ENPP2 (0.51) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL15550064 0.88 ENPP2 (0.51) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL15549996 0.88 ENPP2 (0.66) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL17045096 0.88 ENPP2 (0.66) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL17053656 0.86 ALDH1A1 (0.43) ENPP2ALDH1A1MAPTHPGDKDM2B
SCHEMBL17057704 0.86 ENPP2 (0.52) ENPP2LPAR1ALDH1A1MAPTHPGD
SCHEMBL15553172 0.82 ENPP2 (0.45) ENPP2LPAR1SCN9ARORCAPP
SCHEMBL15553173 0.82 ENPP2 (0.45) ENPP2LPAR1SCN9ARORCAPP
SCHEMBL15550551 0.81 APP (0.46) ENPP2KDM2BCYP2A6APPCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2877185-B1 2-(1-(1-(6-((CYCLOHEXYL)OXY)-5-(TRIFLUOROMETHYL)NAPHTHALEN-2-YL)ETHYL)PIPERIDIN-3-YL)ACETIC ACID DERIVATIVES AS AUTOTAXIN (ATX) MODULATORS FOR THE TREATMENT OF INFLAMMATIONS AND AUTOIMMUNE DISORDERS BIOGEN MA INC (US) 2018-05-23 EP disclosed