SCHEMBL20171876

SCHEMBL20171876

Fc1nc(N2CCCC2)c2nc[nH]c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.41
MAPK1 P28482 3/20 0.41
TP53 P04637 1/20 0.41
IP6K1 Q92551 5/20 0.40
LMNA P02545 2/20 0.40
ALOX15 P16050 1/20 0.40
AKT2 P31751 1/20 0.40
MAP3K5 Q99683 1/20 0.40
JAK3 P52333 2/20 0.36
ADORA3 P0DMS8 5/20 0.36
ADORA2A P29274 5/20 0.36
ADORA1 P30542 4/20 0.36
ADORA2B P29275 1/20 0.35
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20093537 0.86 HRH4 (0.45) HTTMAPK1ADORA3ADORA2AADORA1
SCHEMBL8830247 0.81 CHUK (0.48) HTTMAPK1TP53IP6K1LMNA
SCHEMBL2229901 0.81 NPY5R (0.43) HTTMAPK1TP53LMNAALOX15
SCHEMBL14183741 0.81 HTT (0.41) HTTMAPK1TP53IP6K1LMNA
SCHEMBL4513985 0.80 TLR7 (0.47) HTTMAPK1TP53IP6K1LMNA
SCHEMBL16211583 0.80 CNR2 (0.43)
SCHEMBL14183776 0.80 ABCB1 (0.46) HTTMAPK1TP53LMNAALOX15
SCHEMBL14183739 0.79 ADORA3 (0.42) HTTMAPK1TP53IP6K1LMNA
SCHEMBL14071956 0.79 NPY5R (0.46) HTTMAPK1TP53LMNAALOX15
SCHEMBL8830437 0.79 CHUK (0.50) HTTMAPK1TP53IP6K1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991987-B1 PURINE DERIVATIVES AS CB2 RECEPTOR AGONISTS HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed