SCHEMBL20172003

SCHEMBL20172003

N#Cc1ccc(Nc2ncc(C#CCCCN)c(N)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
SYK P43405 2/20 0.48
KCNH2 Q12809 2/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
FLT3 P36888 1/20 0.41
AURKA O14965 1/20 0.40
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
GRM5 P41594 2/20 0.38
MAOB P27338 1/20 0.38
KDR P35968 3/20 0.38
ABCC3 O15438 1/20 0.38
ESR1 P03372 1/20 0.38
PGR P06401 1/20 0.38
CHRM2 P08172 1/20 0.38
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20172049 0.91 NPC1 (0.53) NPC1RAB9ASYKKCNH2SCN5A
SCHEMBL15584301 0.86 SYK (0.51) NPC1RAB9ASYKFLT3AURKA
SCHEMBL20172050 0.86 SYK (0.51) NPC1RAB9ASYKFLT3AURKA
SCHEMBL16450162 0.84 SYK (0.58) NPC1RAB9ASYKFLT3AURKA
SCHEMBL20172004 0.83 SYK (0.48) NPC1RAB9ASYKKCNH2SCN5A
SCHEMBL15584691 0.82 SYK (0.42) NPC1RAB9ASYKKCNH2SCN5A
SCHEMBL15585199 0.82 FLT3 (0.58) SYKFLT3CHEK1STK17BSTK17A
Hydrochloric Acid SCHEMBL21046222 0.81 FLT3 (0.57) SYKFLT3CHEK1STK17BSTK17A
SCHEMBL15585214 0.79 SYK (0.52) NPC1RAB9ASYKFLT3AURKA
SCHEMBL20172044 0.76 FLT3 (0.54) NPC1RAB9ASYKFLT3AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323811-A1 PRODUCTION METHOD FOR NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND INTERMEDIATE OF SAID NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM Corporation (JP) 2018-05-23 EP disclosed