SCHEMBL20172004

SCHEMBL20172004

N#Cc1ccc(Nc2ncc(C#CCCCN)cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.48
KCNH2 Q12809 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
TDO2 P48775 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRM5 P41594 2/20 0.37
MAOB P27338 1/20 0.37
CHEK1 O14757 2/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20977474 0.84 SYK (0.47) SYKKCNH2SCN5ASCN9ATDO2
SCHEMBL20172003 0.83 NPC1 (0.53) SYKKCNH2SCN5ASCN9AGRM5
SCHEMBL15584301 0.81 SYK (0.51) SYKCHEK1MAPK9MAPK10NPC1
SCHEMBL20172050 0.81 SYK (0.51) SYKCHEK1MAPK9MAPK10NPC1
SCHEMBL16450162 0.79 SYK (0.58) SYKCHEK1MAPK9MAPK10NPC1
SCHEMBL15585199 0.77 FLT3 (0.58) SYKCHEK1STK17BSTK17A
SCHEMBL15584691 0.77 SYK (0.42) SYKKCNH2SCN5ASCN9AGRM5
Hydrochloric Acid SCHEMBL21046222 0.77 FLT3 (0.57) SYKCHEK1STK17BSTK17A
Hydrochloric Acid SCHEMBL7420508 0.76 LOXL2 (0.45) ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL15585214 0.74 SYK (0.52) SYKNPC1RAB9ASTK17BSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323811-A1 PRODUCTION METHOD FOR NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND INTERMEDIATE OF SAID NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM Corporation (JP) 2018-05-23 EP disclosed