SCHEMBL20172469

SCHEMBL20172469

Clc1ccc(Nc2cccnc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.62
MEN1 O00255 4/20 0.62
RAB9A P51151 1/20 0.62
NAMPT P43490 1/20 0.57
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56
NPC1 O15118 1/20 0.55
MAPT P10636 4/20 0.51
LMNA P02545 3/20 0.50
ALDH1A1 P00352 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GAA P10253 1/20 0.50
GFER P55789 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
KIF11 P52732 1/20 0.49
CNR1 P21554 1/20 0.48
CYP17A1 P05093 1/20 0.48
CYP19A1 P11511 1/20 0.47
FLT1 P17948 1/20 0.47
FFAR2 O15552 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14433854 0.90 SCN9A (0.60) KMT2AMEN1RAB9ANAMPTCYP11B1
SCHEMBL1368828 0.85 KIF11 (0.60) KMT2ARAB9ANPC1MAPTLMNA
SCHEMBL29793056 0.85 KIF11 (0.60) KMT2ARAB9ANPC1MAPTLMNA
SCHEMBL4591751 0.83 KMT2A (0.61) KMT2AMEN1RAB9ANAMPTNPC1
SCHEMBL29845262 0.83 KMT2A (0.61) KMT2AMEN1RAB9ANAMPTNPC1
SCHEMBL20194707 0.81 KIF11 (0.53) KMT2AMEN1RAB9ANPC1MAPT
SCHEMBL3954788 0.81 ABL1 (0.58) KMT2AMEN1NPC1MAPTLMNA
SCHEMBL968252 0.80 CYP11B1 (0.56) KMT2AMEN1RAB9ACYP11B1CYP11B2
SCHEMBL11875326 0.80 MAPT (0.55) KMT2AMEN1RAB9ANPC1MAPT
SCHEMBL6431980 0.80 RAB9A (0.62) KMT2ARAB9ANAMPTNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3137459-B1 MORPHOLIN-PYRIDINE DERIVATIVES HAVING AFFINITY TO THE TAAR1 RECEPTOR HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed